Indirect C—H Azidation of Heterocycles via Copper-Catalyzed Regioselective Fragmentation of Unsymmetrical λ3-Iodanes

ChemInform 2013
Dmitrijs Lubriks, Igors Sokolovs, Edgars Sūna

A convenient approach to the synthesis of heteroaryl-substituted azides via C—H activation is followed by direct 1,3-dipolar Cu-catalyzed cycloaddition with terminal alkynes or by direct Cu-catalyzed reductive fragmentation to amino compounds.

Keywords
pyrrole derivatives; fused pyrrole derivatives; triazole derivatives; indole derivatives, isoindole derivatives
DOI
10.1002/chin.201309121
Hyperlink
http://dx.doi.org/10.1002/chin.201309121

Lubriks, D., Sokolovs, I., Sūna, E. Indirect C—H Azidation of Heterocycles via Copper-Catalyzed Regioselective Fragmentation of Unsymmetrical λ3-Iodanes. ChemInform, 2013, Vol.44, Iss.9, pp.121-121. ISSN 1522-2667. Available from: doi:10.1002/chin.201309121

Publication language
English (en)