RTU Research Outputs and Resources: Reasearch Staff

Information about Author

Name, Surname:

Raivis Žalubovskis

Department:

(14A24) Bioloģiski aktīvo savienojumu ķīmijas tehnoloģijas katedra

Scientific Degree:

Doktors

E-mail:

Raivis.Zalubovskis(at)rtu.lv

Publications

42 items found, displaying 1 to 10.

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors
(2021)

Andrea Angeli, Fabrizio Carta, Alessio Nocentini, Jean-Yves Winum, Raivis Žalubovskis, valentina Onnis, Wagdy E. Eldehna, Clemente Capasso, Simone Carradori, William A. Donald, Shoukat Dedhar, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Reconsidering Anion Inhibitors in the General Context of Drug Design Studies of Modulators of Activity of the Classical Enzyme Carbonic Anhydrase
(2021)

A Nocentini, A Angeli, F Carta, J.-Y Winum, Raivis Žalubovskis, S Carradori, C Capasso, W.A Donald, C.T Supuran
Scientific article indexed in SCOPUS or WOS database

Base-Free Catalytic Wittig-/Cross-Coupling Reaction Sequence as Short Synthetic Strategy for the Preparation of Highly Functionalized Arylbenzoxepinones
(2021)

L Pudnika, I Domraceva, T Werner, Raivis Žalubovskis, A Grandane
Scientific article indexed in SCOPUS or WOS database

Aryl Derivatives of 3H-1,2-benzoxathiepine 2,2-Dioxide as Carbonic Anhydrase Inhibitors
(2020)

Aleksandrs Pustenko, A. Nocentini, A. Alafeefy, A. Balašova, M. Krasavin, Raivis Žalubovskis, C.T. Supuran
Scientific article indexed in SCOPUS or WOS database

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment
(2020)

Andrea Angeli, Fabrizio Carta, Alessio Nocentini, Jean-Yves Winum, Raivis Žalubovskis, Atilla Akdemir, valentina Onnis, Wagdy E. Eldehna, Clemente Capasso, Giuseppina De Simone, Simona Maria Monti, Simone Carradori, William A. Donald, Shoukat Dedhar, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Development of Oxathiino[6,5-b]pyridine 2,2-Dioxide Derivatives as Selective Inhibitors of Tumor-Related Carbonic Anhydrases IX and XII
(2020)

Aiga Grandane, Alessio Nocentini, Ilona Domračeva, Raivis Žalubovskis, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors
(2020)

Aiga Grandane, Alessio Nocentini, Thomas Werner, Raivis Žalubovskis, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Further Exploration of DVD-445 as a Lead Thioredoxin Reductase (TrxR) Inhibitor for Cancer Therapy: Optimization of Potency and Evaluation of Anticancer Potential
(2020)

Mirna Jovanovic, Daniil Zhukovsky, Ana Podolski-Renic, Raivis Žalubovskis, Dmitry Dar`in, Vladimir Sharoyko, Tatiana Tennikova, Milica Pešic, Mikhail Krasavin
Scientific article indexed in SCOPUS or WOS database

7-Acylamino-3H-1,2-benzoxathiepine 2,2-Dioxides as New Isoform-Selective Carbonic Anhydrase IX and XII Inhibitors
(2020)

Aleksandrs Pustenko, Alessio Nocentini, Anastasija Balašova, Mikhail Krasavin, Raivis Žalubovskis, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Sulfocoumarins as Dual Inhibitors of Human Carbonic Anhydrase Isoforms IX/XII and of Human Thioredoxin Reductase
(2020)

Mikhail Krasavin, Raivis Žalubovskis, Aiga Grandane, Ilona Domračeva, Petr Zhmurov, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Information about Author

Publications

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors
(2021)

Reconsidering Anion Inhibitors in the General Context of Drug Design Studies of Modulators of Activity of the Classical Enzyme Carbonic Anhydrase
(2021)

Base-Free Catalytic Wittig-/Cross-Coupling Reaction Sequence as Short Synthetic Strategy for the Preparation of Highly Functionalized Arylbenzoxepinones
(2021)

Aryl Derivatives of 3H-1,2-benzoxathiepine 2,2-Dioxide as Carbonic Anhydrase Inhibitors
(2020)

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment
(2020)

Development of Oxathiino[6,5-b]pyridine 2,2-Dioxide Derivatives as Selective Inhibitors of Tumor-Related Carbonic Anhydrases IX and XII
(2020)

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors
(2020)

Further Exploration of DVD-445 as a Lead Thioredoxin Reductase (TrxR) Inhibitor for Cancer Therapy: Optimization of Potency and Evaluation of Anticancer Potential
(2020)

7-Acylamino-3H-1,2-benzoxathiepine 2,2-Dioxides as New Isoform-Selective Carbonic Anhydrase IX and XII Inhibitors
(2020)

Sulfocoumarins as Dual Inhibitors of Human Carbonic Anhydrase Isoforms IX/XII and of Human Thioredoxin Reductase
(2020)

Supervised Dissertations

Synthesis of a New Type of Carbonic Anhydrases Inhibitors
(2020)

Synthesis of the Inhibitors of Carbonic Anhydrases and Thioredoxin Reductase as Potential Anticancer Agents
(2017)

Information about Author

Publications

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors (2021)

Reconsidering Anion Inhibitors in the General Context of Drug Design Studies of Modulators of Activity of the Classical Enzyme Carbonic Anhydrase (2021)

Base-Free Catalytic Wittig-/Cross-Coupling Reaction Sequence as Short Synthetic Strategy for the Preparation of Highly Functionalized Arylbenzoxepinones (2021)

Aryl Derivatives of 3H-1,2-benzoxathiepine 2,2-Dioxide as Carbonic Anhydrase Inhibitors (2020)

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment (2020)

Development of Oxathiino[6,5-b]pyridine 2,2-Dioxide Derivatives as Selective Inhibitors of Tumor-Related Carbonic Anhydrases IX and XII (2020)

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors (2020)

Further Exploration of DVD-445 as a Lead Thioredoxin Reductase (TrxR) Inhibitor for Cancer Therapy: Optimization of Potency and Evaluation of Anticancer Potential (2020)

7-Acylamino-3H-1,2-benzoxathiepine 2,2-Dioxides as New Isoform-Selective Carbonic Anhydrase IX and XII Inhibitors (2020)

Sulfocoumarins as Dual Inhibitors of Human Carbonic Anhydrase Isoforms IX/XII and of Human Thioredoxin Reductase (2020)

Supervised Dissertations

Synthesis of a New Type of Carbonic Anhydrases Inhibitors (2020)

Synthesis of the Inhibitors of Carbonic Anhydrases and Thioredoxin Reductase as Potential Anticancer Agents (2017)

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors
(2021)

Reconsidering Anion Inhibitors in the General Context of Drug Design Studies of Modulators of Activity of the Classical Enzyme Carbonic Anhydrase
(2021)

Base-Free Catalytic Wittig-/Cross-Coupling Reaction Sequence as Short Synthetic Strategy for the Preparation of Highly Functionalized Arylbenzoxepinones
(2021)

Aryl Derivatives of 3H-1,2-benzoxathiepine 2,2-Dioxide as Carbonic Anhydrase Inhibitors
(2020)

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment
(2020)

Development of Oxathiino[6,5-b]pyridine 2,2-Dioxide Derivatives as Selective Inhibitors of Tumor-Related Carbonic Anhydrases IX and XII
(2020)

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors
(2020)

Further Exploration of DVD-445 as a Lead Thioredoxin Reductase (TrxR) Inhibitor for Cancer Therapy: Optimization of Potency and Evaluation of Anticancer Potential
(2020)

7-Acylamino-3H-1,2-benzoxathiepine 2,2-Dioxides as New Isoform-Selective Carbonic Anhydrase IX and XII Inhibitors
(2020)

Sulfocoumarins as Dual Inhibitors of Human Carbonic Anhydrase Isoforms IX/XII and of Human Thioredoxin Reductase
(2020)

Synthesis of a New Type of Carbonic Anhydrases Inhibitors
(2020)

Synthesis of the Inhibitors of Carbonic Anhydrases and Thioredoxin Reductase as Potential Anticancer Agents
(2017)