Indirect C—H Azidation of Heterocycles via Copper-Catalyzed Regioselective Fragmentation of Unsymmetrical λ3-Iodanes

ChemInform 2013
Dmitrijs Lubriks, Igors Sokolovs, Edgars Sūna

A convenient approach to the synthesis of heteroaryl-substituted azides via C—H activation is followed by direct 1,3-dipolar Cu-catalyzed cycloaddition with terminal alkynes or by direct Cu-catalyzed reductive fragmentation to amino compounds.

Atslēgas vārdi
pyrrole derivatives; fused pyrrole derivatives; triazole derivatives; indole derivatives, isoindole derivatives
DOI
10.1002/chin.201309121
Hipersaite
http://dx.doi.org/10.1002/chin.201309121

Lubriks, D., Sokolovs, I., Sūna, E. Indirect C—H Azidation of Heterocycles via Copper-Catalyzed Regioselective Fragmentation of Unsymmetrical λ3-Iodanes. ChemInform, 2013, Vol.44, Iss.9, 121.-121.lpp. ISSN 1522-2667. Pieejams: doi:10.1002/chin.201309121

Publikācijas valoda
English (en)