RTU Zinātniskās darbības rezultāti un resursi: Personāls

Structural Basis of Saccharin Derivative Inhibition of Carbonic Anhydrase IX
(2023)

Janis Leitans, Andris Kazaks, Janis Bogans, Claudiu T. Supuran, Ināra Akopjana, Jekaterīna Ivanova, Raivis Žalubovskis, Kaspars Tārs
Zinātniskais raksts, kas indeksēts Web of science un/vai Scopus datu bāzē

Atropo/Tropo Flexibility: A Tool for Design and Synthesis of Self-Adaptable Inhibitors of Carbonic Anhydrases and Their Antiproliferative Effect
(2023)

Jekaterīna Ivanova, Alessio Nocentini, Kaspars Tārs, Janis Leitans, Elviss Dvinskis, Andris Kazaks, Ilova Domračeva, Claudiu T. Supuran, Raivis Žalubovskis
Zinātniskais raksts, kas indeksēts Web of science un/vai Scopus datu bāzē

3H-1,2-Benzoxathiepine 2,2-Dioxides: a New Class of Isoform-Selective Carbonic Anhydrase Inhibitors
(2017)

Aleksandrs Pustenko, Dmitrijs Stepanovs, Raivis Žalubovskis, Daniela Vullo, Andris Kazaks, Janis Leitans, Kaspars Tārs, Claudiu Supuran
Zinātniskais raksts, kas indeksēts Web of science un/vai Scopus datu bāzē

N-Substituted and Ring Opened Saccharin Derivatives Selectively Inhibit Transmembrane, Tumor-Associated Carbonic Anhydrases IX and XII
(2017)

Jekaterīna Ivanova, Fabrizio Carta, Daniela Vullo, Janis Leitans, Andris Kazaks, Kaspars Tārs, Raivis Žalubovskis, Claudiu T. Supuran
Zinātniskais raksts, kas indeksēts Web of science un/vai Scopus datu bāzē

CCDC 1526002: Experimental Crystal Structure Determination
(2017)

Aleksandrs Pustenko, Dmitrijs Stepanovs, Raivis Žalubovskis, Daniela Vullo, Andris Kazaks, Janis Leitans, Kaspars Tārs, Claudiu T. Supuran
Publikācija internetā

5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with Effective Carbonic Anhydrase Inhibitory Activity: Solution and Crystallographic Investigations
(2017)

Jekaterīna Ivanova, Agnese Balode, Raivis Žalubovskis, Janis Leitans, Andris Kazaks, Daniela Vullo, Kaspars Tārs, Claudiu T. Supuran
Zinātniskais raksts, kas indeksēts Web of science un/vai Scopus datu bāzē

Challenging Design and Synthesis of Inhibitors of Carbonic Anhydrases
(2016)

Jekaterīna Ivanova, Agnese Balode, Aleksandrs Pustenko, Raivis Žalubovskis, Aiga Grandane, Ilona Domračeva, Kaspars Tārs, Janis Leitans
Raksts konferenču tēžu krājumā

X-Ray Crystallography-Promoted Drug Design of Carbonic Anhydrase Inhibitors
(2015)

Jekaterīna Ivanova, Raivis Žalubovskis, Muhammet Tanc, Andris Kazaks, Claudiu T. Supuran, Kaspars Tārs, Janis Leitans
Zinātniskais raksts, kas indeksēts Web of science un/vai Scopus datu bāzē

Efficient Expression and Crystallization System of Cancer-Associated Carbonic Anhydrase Isoform IX
(2015)

Jekaterīna Ivanova, Agnese Balode, Raivis Žalubovskis, Kaspars Tārs, Andris Kazaks, Janis Leitans, Claudiu T. Supuran
Zinātniskais raksts, kas indeksēts Web of science un/vai Scopus datu bāzē

Targeting Carnitine Biosynthesis: Discovery of New Inhibitors against γ-Butyrobetaine Hydroxylase
(2014)

Kaspars Tārs, Janis Leitans, Andris Kazaks, Diāna Zeļencova-Gopejenko, Edgars Liepiņš, Jānis Kūka, Marina Makrecka, Daina Lola, Viktors Andrianovs, Daina Gustina, Solveiga Grinberga, Edvards Liepiņš, Ivars Kalviņš, Maija Dambrova, Einārs Loža, Osvalds Pugovičs
Zinātniskais raksts, kas indeksēts Web of science un/vai Scopus datu bāzē

Informācija par autoru

Publikācijas

Structural Basis of Saccharin Derivative Inhibition of Carbonic Anhydrase IX
(2023)

Atropo/Tropo Flexibility: A Tool for Design and Synthesis of Self-Adaptable Inhibitors of Carbonic Anhydrases and Their Antiproliferative Effect
(2023)

3H-1,2-Benzoxathiepine 2,2-Dioxides: a New Class of Isoform-Selective Carbonic Anhydrase Inhibitors
(2017)

N-Substituted and Ring Opened Saccharin Derivatives Selectively Inhibit Transmembrane, Tumor-Associated Carbonic Anhydrases IX and XII
(2017)

CCDC 1526002: Experimental Crystal Structure Determination
(2017)

5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with Effective Carbonic Anhydrase Inhibitory Activity: Solution and Crystallographic Investigations
(2017)

Challenging Design and Synthesis of Inhibitors of Carbonic Anhydrases
(2016)

X-Ray Crystallography-Promoted Drug Design of Carbonic Anhydrase Inhibitors
(2015)

Efficient Expression and Crystallization System of Cancer-Associated Carbonic Anhydrase Isoform IX
(2015)

Targeting Carnitine Biosynthesis: Discovery of New Inhibitors against γ-Butyrobetaine Hydroxylase
(2014)

Informācija par autoru

Publikācijas

Structural Basis of Saccharin Derivative Inhibition of Carbonic Anhydrase IX (2023)

Atropo/Tropo Flexibility: A Tool for Design and Synthesis of Self-Adaptable Inhibitors of Carbonic Anhydrases and Their Antiproliferative Effect (2023)

3H-1,2-Benzoxathiepine 2,2-Dioxides: a New Class of Isoform-Selective Carbonic Anhydrase Inhibitors (2017)

N-Substituted and Ring Opened Saccharin Derivatives Selectively Inhibit Transmembrane, Tumor-Associated Carbonic Anhydrases IX and XII (2017)

CCDC 1526002: Experimental Crystal Structure Determination (2017)

5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with Effective Carbonic Anhydrase Inhibitory Activity: Solution and Crystallographic Investigations (2017)

Challenging Design and Synthesis of Inhibitors of Carbonic Anhydrases (2016)

X-Ray Crystallography-Promoted Drug Design of Carbonic Anhydrase Inhibitors (2015)

Efficient Expression and Crystallization System of Cancer-Associated Carbonic Anhydrase Isoform IX (2015)

Targeting Carnitine Biosynthesis: Discovery of New Inhibitors against γ-Butyrobetaine Hydroxylase (2014)

Structural Basis of Saccharin Derivative Inhibition of Carbonic Anhydrase IX
(2023)

Atropo/Tropo Flexibility: A Tool for Design and Synthesis of Self-Adaptable Inhibitors of Carbonic Anhydrases and Their Antiproliferative Effect
(2023)

3H-1,2-Benzoxathiepine 2,2-Dioxides: a New Class of Isoform-Selective Carbonic Anhydrase Inhibitors
(2017)

N-Substituted and Ring Opened Saccharin Derivatives Selectively Inhibit Transmembrane, Tumor-Associated Carbonic Anhydrases IX and XII
(2017)

CCDC 1526002: Experimental Crystal Structure Determination
(2017)

5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with Effective Carbonic Anhydrase Inhibitory Activity: Solution and Crystallographic Investigations
(2017)

Challenging Design and Synthesis of Inhibitors of Carbonic Anhydrases
(2016)

X-Ray Crystallography-Promoted Drug Design of Carbonic Anhydrase Inhibitors
(2015)

Efficient Expression and Crystallization System of Cancer-Associated Carbonic Anhydrase Isoform IX
(2015)

Targeting Carnitine Biosynthesis: Discovery of New Inhibitors against γ-Butyrobetaine Hydroxylase
(2014)